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TargetMol | Compound Library

抗糖尿病库现货

Anti-Diabetic Compound Library

产品编号 L1900

糖尿病是一种以高血糖为特征的代谢性疾病,长期的高血糖会导致全身各种组织功能障碍,如果出现并发症,糖尿病会对生活质量产生重大影响,并可能降低预期寿命,目前仍然无法治愈糖尿病,只能通过饮食调节和药物辅助治疗进行病情控制。 TargetMol 抗糖尿病库包含了 683 个糖尿病相关活性化合物,是研究糖尿病的优良工具和药物筛选的极佳载体。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L1900

抗糖尿病库
规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 683种生物活性小分子化合物;
  • 靶点包括SGLT、PPAR、DPP-4、OC receptor、AMPK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库定制

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Library Customization | TargetMol 化合物库组成

PPAR
Autophagy
NF-κB
Apoptosis
AMPK
mTOR
GSK-3
Endogenous Metabolite
JNK
PI3K
Antibacterial
Sirtuin
COX
Potassium Channel
DPP-4
Proteasome
Akt
TNF
Ferroptosis
CDK
Glucagon Receptor
SGLT
STAT
GPR
Antibiotic
ERK
P450
DNA-PK
Mitophagy
p38 MAPK
Calcium Channel
Wnt/beta-catenin
Parasite
Glucosidase
Reactive Oxygen Species
IL Receptor
Influenza Virus
RAAS
Caspase
Antifungal
PARP
Prostaglandin Receptor
MMP
transporter
5-HT Receptor
Cannabinoid Receptor
S6 Kinase
Dehydrogenase
Lipoxygenase
IκB/IKK
ATM/ATR
Beta Amyloid
HIV Protease
ATPase
Src
Reductase
Phosphatase
Virus Protease
PKC
IRE1
PDE
DNA/RNA Synthesis
Nrf2
HDAC
FLT
Sodium Channel
Tyrosinase
p53
NO Synthase
Histone Methyltransferase
NADPH
Glucokinase
VEGFR
TRP/TRPV Channel
Glucocorticoid Receptor
SIK
E1/E2/E3 Enzyme
Mitochondrial Metabolism
BCL
JAK
HSV
Epigenetic Reader Domain
MAPK
AChE
AChR
BACE
PKA
HBV
ROCK
Adrenergic Receptor
Endothelin Receptor
IGF-1R
Interleukin
EGFR
TLR
Casein Kinase
GABA Receptor
MEK
FGFR
Thrombin
HIF/HIF Prolyl-Hydroxylase
NOS
Carbonic Anhydrase
Dopamine Receptor
Integrin
Antioxidant
Adenosine Receptor
Histamine Receptor
Glutathione Peroxidase
ABC
Estrogen Receptor/ERR
Rho
Serine Protease
FXR
Leukotriene Receptor
Topoisomerase
Drug Metabolite
ROS
Fatty Acid Synthase
PDGFR
CCR
Vasopressin Receptor
Chk
Epoxide Hydrolase
Aurora Kinase
Norepinephrine
DNA
Androgen Receptor
TGF-beta/Smad
SARS-CoV
Retinoid Receptor
Phospholipase
HIF
c-RET
NOD
NADPH-oxidase
Sigma receptor
Microtubule Associated
CFTR
Thyroid hormone receptor(THR)
advanced glycation end products
Chloride channel
NPC1L1
Estrogen/progestogen Receptor
YAP
LTR
Histone Demethylase
PERK
Tie-2
Tyrosine Kinases
Serotonin Transporter
Cysteine Protease
Liver X Receptor
Amylase
Aryl Hydrocarbon Receptor
MAO
Annexin A
FLAP
LDL
Raf
Phosphorylase
Antifection
Hexokinase
Guanylate cyclase
Opioid Receptor
PROTAC Linker
PAK
Bombesin Receptor
PGC-1α
CXCR
OX Receptor
GluR
CaMK
ATP Citrate Lyase
Beta-Secretase
PGE Synthase
P-gp
OAT
Trk receptor
GPCR19
Free radical scavengers
ASK
PAI-1
ALK
Carboxypeptidase
Reverse Transcriptase
c-Fms
Aromatase
PI4K
PDK
c-Kit
IRAK
HMG-CoA Reductase
AhR
NOD-like Receptor (NLR)
Monoamine Oxidase

Keywords