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TargetMol | Compound Library

抗肥胖化合物库现货

Anti-Obesity Compound Library

产品编号 L7100

近年来肥胖已成为全球普遍的公共健康问题,肥胖是一种由多种因素(遗传、饮食习惯、生活方式和环境)相互作用引起的复杂的疾病,通常伴随着胰岛素抵抗、氧化应激和炎症标志物表达增加,导致体内脂肪含量增加。肥胖容易引起糖尿病,高血压,动脉硬化等多种代谢紊乱性疾病。肥胖管理的基本策略(如饮食控制、体育运动、手术治疗)分别具有不同程度的局限性和副作用。因此,许多研究人员试图从食物或药物中寻找出抗肥胖的生物活性成分,特别是抑制脂肪等高能量物质吸收过程的化合物、促进脂肪分解的化合物、增加机体代谢能量消耗的化合物,这些化合物包括:脂肪酶抑制剂、a-葡萄糖苷酶抑制剂、麦芽糖酶抑制剂等。 随着经济发展,肥胖问题已成为全球面临的严峻问题,所以科学家对肥胖的关注和研究更是有增无减。通过对文献和公开资料的整理,我们精心筛选了2247 个抗肥胖化合物组成抗肥胖化合物库,适合于抗肥胖的相关研究。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L7100

抗肥胖化合物库
规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2247个抗肥胖化合物的独特集合,可用于高通量筛选和高内涵筛选;
  • 提供产品的来源、化学信息和生物学信息,为筛选提供理论方向和研究基础;
  • 结构多样,药效显著,可渗透细胞;
  • NMR和HPLC技术保证产品高纯度。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
PI3K
Reactive Oxygen Species
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
PPAR
mTOR
ERK
p38 MAPK
Akt
Antibacterial
NF-κB
Histamine Receptor
Dopamine Receptor
AMPK
Raf
GSK-3
Ras
COX
Wnt/beta-catenin
JNK
VEGFR
ROS
MAPK
CDK
MEK
Phospholipase
JAK
Lipoxygenase
AChR
PKA
DNA-PK
Parasite
TGF-beta/Smad
Nrf2
TNF
Ferroptosis
Influenza Virus
S6 Kinase
Antifungal
Prostaglandin Receptor
P450
Antioxidant
Src
PKC
Fatty Acid Synthase
PDGFR
Antibiotic
GPR
ALK
Potassium Channel
ATM/ATR
Caspase
IL Receptor
HIV Protease
FLT
Mitophagy
Calcium Channel
STAT
PDE
FAAH
Dehydrogenase
c-Kit
Adenosine Receptor
Serotonin Transporter
Norepinephrine
PDK
Cannabinoid Receptor
Virus Protease
Opioid Receptor
Hedgehog/Smoothened
MMP
DNA/RNA Synthesis
Casein Kinase
FGFR
Aurora Kinase
PI4K
Lipase
PARP
NO Synthase
Tyrosine Kinases
SGLT
Rho
Glucagon Receptor
AChE
Transferase
ROCK
BCL
c-RET
Estrogen/progestogen Receptor
Stearoyl-CoA Desaturase (SCD)
EGFR
transporter
Acetyl-CoA Carboxylase
HIF/HIF Prolyl-Hydroxylase
c-Met/HGFR
TRP/TRPV Channel
Bcr-Abl
Mitochondrial Metabolism
CaMK
IκB/IKK
Tyrosinase
Smo
CXCR
Interleukin
Trk receptor
ROS Kinase
MLK
Glucosidase
Chk
IGF-1R
P-gp
HDAC
Melanocortin Receptor
NOS
LPL Receptor
DYRK
Phosphatase
Glucocorticoid Receptor
SIK
Topoisomerase
HSV
OX Receptor
MNK
GABA Receptor
Sodium Channel
S1P Receptor
P2Y Receptor
CETP
HBV
Serine/threonin kinase
PAFR
Drug Metabolite
PTEN
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Acyltransferase
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Syk
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ATPase
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MAO
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SARS-CoV
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ASK
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FAK
HER
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NPC1L1
HCV Protease
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PERK
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TOPK
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Pim
Aryl Hydrocarbon Receptor
iGluR
LDL
GluR
cAMP
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TLR
GPCR19
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p53
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BACE
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ABC
MRP
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Adiponectin receptor
UGT
GRK
MAGL
Neuropeptide Y Receptor
ATP Citrate Lyase
PGE Synthase
HSP
Reverse Transcriptase
Retinoid Receptor
KLF
PLK
cholecystokinin
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
Proteasome
Monocarboxylate transporter
ROR
YAP
RAR/RXR 
Tie-2
c-Myc
CaSR
GNRH Receptor
Cysteine Protease
Immunology/Inflammation related
IAP
CSF-1R
E1/E2/E3 Enzyme
RIP kinase
Gamma-secretase
MT Receptor
Guanylate cyclase
DNA Alkylation
PAK
ACK
DNA
Androgen Receptor
Lipid
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RSV
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Progesterone Receptor
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PYK2
FLAP
NMDAR
BTK
Monoamine Transporter
DPP-4
PGC-1α
CCR
Bradykinin Receptor
Somatostatin
PAD
Epoxide Hydrolase
OXPHOS
BCRP
Glutathione reductase
STING
Histone Acetyltransferase
PAI-1
Hippo pathway
GPX
ribosome
LPA Receptor
Oxytocin Receptor
Hydroxylase
RXFP receptor
DAPK
Discoidin Domain Receptor (DDR)
Gap Junction Protein
Platelet aggregation
NOD
BMI-1
DNA Methyltransferase
IRAK
Thrombin
lysosomal autophagy
AhR
CFTR
Imidazoline Receptor
PD-1/PD-L1
Kinesin

Keywords