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TargetMol | Compound Library

离子通道库现货

Ion Channel Inhibitor Library

产品编号 L2300

离子跨膜通道的调节是治疗多种疾病的基础,离子通道是开发新的高效药物治疗的重要靶点,随着人类基因组计划的完成和转录机制研究的深入,离子通道分布的组织特异性逐渐得以阐明,这将使离子通道成为一类有选择性的组织特异性药物靶点。离子通道对于细胞间通讯至关重要,并调节多种重要的生理过程,这些过程功能障碍,可导致广泛的疾病和病理状况,如糖尿病、神经性疼痛、心血管疾病、大脑和外周血管疾病、哮喘、神经退行性疾病。 为满足客户离子通道相关研究的化合物需求,我们根据文献报道和其他公开资料精心整理 1147 种与离子通道相关的生物活性小分子化合物,适用于离子通道相关的疾病和药物研究。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L2300

离子通道库
规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1147种与离子通道相关的生物活性小分子化合物的特有集合,用于离子通道相关的疾病和药物研究,可用于高通量筛选和高内涵筛选;
  • 靶点含K+通道、Ca2+通道、Na+通道、质子泵等;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;
  • 其中一些活性化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Calcium Channel
Calcium Channel
Potassium Channel
Potassium Channel
Sodium Channel
Sodium Channel
GABA Receptor
GABA Receptor
TRP/TRPV Channel
TRP/TRPV Channel
AChR
AChR
iGluR
iGluR
Autophagy
Autophagy
Endogenous Metabolite
Endogenous Metabolite
NMDAR
NMDAR
P2X Receptor
P2X Receptor
Apoptosis
Apoptosis
Chloride channel
Chloride channel
5-HT Receptor
5-HT Receptor
Parasite
Parasite
GluR
GluR
Antibacterial
Antibacterial
Adrenergic Receptor
Adrenergic Receptor
NF-κB
NF-κB
P450
P450
Dopamine Receptor
COX
Dopamine Receptor
COX
HER
Histamine Receptor
Histamine Receptor
HER
Reactive Oxygen Species
Reactive Oxygen Species
HIV Protease
HIV Protease
Antibiotic
ATPase
PPAR
PPAR
ATPase
Antibiotic
TNF
TNF
EGFR
P-gp
Cannabinoid Receptor
Carbonic Anhydrase
AChE
Cannabinoid Receptor
AChE
Carbonic Anhydrase
EGFR
P-gp
Ferroptosis
PKC
SARS-CoV
IL Receptor
VDAC
ABC
ERK
DNA/RNA Synthesis
PDE
CaMK
PKC
SARS-CoV
ABC
ERK
CaMK
DNA/RNA Synthesis
PDE
VDAC
IL Receptor
Ferroptosis
Antioxidant
Drug Metabolite
GPR
Lipoxygenase
HCN Channel
Topoisomerase
PKA
Mitophagy
MRP
Na+/Ca2+ Exchanger
Anti-infection
Influenza Virus
Virus Protease
Lipoxygenase
Mitophagy
MRP
Na+/Ca2+ Exchanger
Anti-infection
Influenza Virus
Virus Protease
PKA
HCN Channel
Topoisomerase
Antioxidant
Drug Metabolite
GPR
Monoamine Transporter
NO Synthase
PAFR
Serine/threonin kinase
Norepinephrine
HDAC
Phospholipase
AMPK
Caspase
HMG-CoA Reductase
NADPH
RAAS
Antifungal
LDL
Transaminase
AMPK
Caspase
HMG-CoA Reductase
NADPH
Antifungal
LDL
Transaminase
HDAC
Phospholipase
RAAS
Norepinephrine
Monoamine Transporter
NO Synthase
PAFR
Serine/threonin kinase
NOD
TGF-beta/Smad
cAMP
Dehydrogenase
HSV
Mitochondrial Metabolism
MT Receptor
ROCK
Wnt/beta-catenin
mTOR
Acyltransferase
Gamma-secretase
Interleukin
NOS
AhR
Beta Amyloid
DNA Methyltransferase
HBV
transporter
Beta-Secretase
HCV Protease
IκB/IKK
MEK
STAT
Antifection
GluCls
Opioid Receptor
Tyrosinase
cAMP
Dehydrogenase
HSV
Mitochondrial Metabolism
MT Receptor
ROCK
AhR
Beta Amyloid
DNA Methyltransferase
HBV
Antifection
GluCls
Opioid Receptor
Wnt/beta-catenin
Tyrosinase
Beta-Secretase
HCV Protease
IκB/IKK
MEK
STAT
Acyltransferase
Gamma-secretase
Interleukin
NOS
transporter
mTOR
NOD
TGF-beta/Smad
CFTR
Gap Junction Protein
GSK-3
GST
p38 MAPK
PAI-1
S1P Receptor
CSF-1R
GlyT
Monocarboxylate transporter
NOD-like Receptor (NLR)
Platelet aggregation
Proton pump
Transferase
UGT
BCL
DNA
LPL Receptor
N-Acetylglucosaminyltransferase
PARP
Prostaglandin Receptor
Reductase
Trk receptor
Akt
BCRP
FXR
Microtubule Associated
Sigma receptor
VEGFR
DNA gyrase
IGF-1R
MAO
PAK
Piezo Channel
Src
Integrin
JNK
Na-K-Cl cotransporter
Proteasome
Androgen Receptor
Anion Exchanger
Arrestin
CDK
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
Glucocorticoid Receptor
LTR
Phosphatase
PKM
Protease-activated Receptor
ROS
Serotonin Transporter
Thrombin
CSF-1R
GlyT
Monocarboxylate transporter
NOD-like Receptor (NLR)
Platelet aggregation
Proton pump
DNA gyrase
IGF-1R
MAO
PAK
Piezo Channel
Androgen Receptor
Anion Exchanger
Arrestin
CDK
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
Glucocorticoid Receptor
LTR
Phosphatase
PKM
Protease-activated Receptor
ROS
Serotonin Transporter
Transferase
UGT
Thrombin
Integrin
JNK
Na-K-Cl cotransporter
Proteasome
Akt
BCRP
FXR
Microtubule Associated
Src
Sigma receptor
VEGFR
BCL
DNA
LPL Receptor
N-Acetylglucosaminyltransferase
PARP
Prostaglandin Receptor
Reductase
Trk receptor
CFTR
Gap Junction Protein
GSK-3
GST
p38 MAPK
PAI-1
S1P Receptor