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Islatravir (MK-8591) 是一种核苷逆转录酶抑制剂,是抗HIV-1药物,对 HIV-1 (WT),HIV-1 (M184V),HIV-1 (MDR) 的EC50值分别为 0.068 nM,3.1 nM 和 0.15 nM。
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Islatravir (MK-8591) 是一种核苷逆转录酶抑制剂,是抗HIV-1药物,对 HIV-1 (WT),HIV-1 (M184V),HIV-1 (MDR) 的EC50值分别为 0.068 nM,3.1 nM 和 0.15 nM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 997 | 现货 | |
5 mg | ¥ 2,660 | 现货 | |
10 mg | ¥ 3,730 | 现货 | |
25 mg | ¥ 6,390 | 现货 | |
50 mg | ¥ 8,280 | 现货 | |
100 mg | ¥ 10,900 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 2,920 | 现货 |
产品描述 | Islatravir (MK-8591) is an effective anti-HIV-1 agent. It acts as a nucleoside reverse transcriptase inhibitor (EC50s: 0.068 nM, 3.1 nM, and 0.15 nM for HIV-1 (WT), HIV-1 (M184V), HIV-1 (MDR), respectively). |
靶点活性 | HIV-1 (MDR):0.15 nM (EC50), HIV-1 (M184V):3.1 nM (EC50), HIV-1 (WT):0.068 nM (EC50) |
别名 | MK-8591 |
分子量 | 293.25 |
分子式 | C12H12FN5O3 |
CAS No. | 865363-93-5 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||||||||||||
溶解度信息 | H2O: 3 mg/mL (10.23 mM), Sonication and heating to 60℃ are recommended. DMSO: 100 mg/mL (341.01 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||||||||||||||||||||||
H2O/DMSO
DMSO
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