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EP2 receptor antagonist-2 (CID891729)为EP2受体拮抗剂,能够抑制PGE2诱导的EP2受体激活,并阻断由N-甲基-D-天冬氨酸(NMDA)引起的乳酸脱氢酶(LDH)释放。
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EP2 receptor antagonist-2 (CID891729)为EP2受体拮抗剂,能够抑制PGE2诱导的EP2受体激活,并阻断由N-甲基-D-天冬氨酸(NMDA)引起的乳酸脱氢酶(LDH)释放。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 428 | 现货 | |
5 mg | ¥ 995 | 现货 | |
10 mg | ¥ 1,660 | 现货 | |
25 mg | ¥ 3,360 | 现货 | |
50 mg | ¥ 4,900 | 现货 | |
100 mg | ¥ 6,980 | 现货 | |
500 mg | ¥ 13,900 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 1,130 | 现货 |
产品描述 | EP2 receptor antagonist-2 (CID891729) is a compound that not only serves as an antagonist to the EP2 receptor, blocking its activation by PGE2, but also reduces lactate dehydrogenase (LDH) release triggered by N-methyl-D-aspartate (NMDA). |
分子量 | 309.29 |
分子式 | C15H14F3N3O |
CAS No. | 615273-95-5 |
存储 | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 112.5 mg/mL (363.7 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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