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QS11 是一种ARFGAP1抑制剂(EC50:1.5 µM)。QS 11 能抑制 ARFGAP 过表达的乳腺癌细胞迁移。QS 11 通过影响蛋白质运输来增强 Wnt/β-catenin 信号。
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QS11 是一种ARFGAP1抑制剂(EC50:1.5 µM)。QS 11 能抑制 ARFGAP 过表达的乳腺癌细胞迁移。QS 11 通过影响蛋白质运输来增强 Wnt/β-catenin 信号。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 319 | 现货 | |
2 mg | ¥ 457 | 现货 | |
5 mg | ¥ 818 | 现货 | |
10 mg | ¥ 1,320 | 现货 | |
25 mg | ¥ 2,650 | 现货 | |
50 mg | ¥ 3,980 | 现货 | |
100 mg | ¥ 5,970 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 987 | 现货 |
产品描述 | QS11 is a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor. Modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling pathway to upregulate β-catenin nuclear translocation. Also reduces in vitro migration of metastatic human breast cancer cells. |
靶点活性 | ARFGAP1:1.5 µM (EC50) |
别名 | QS 11 |
分子量 | 567.68 |
分子式 | C36H33N5O2 |
CAS No. | 944328-88-5 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||||||||||||
溶解度信息 | Ethanol: 100 mM DMSO: 55 mg/mL (96.88 mM) | ||||||||||||||||||||||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||||||||||||||||||||||
DMSO/Ethanol
Ethanol
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