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TAO Kinase inhibitor 1 是一种ATP 竞争性的thousand-and-one amino acid kinases (TAOK)选择性抑制剂,对于 TAOK1 和 TAOK2 的IC50s 分别为 11 nM 和 15 nM。它能够延迟有丝分裂以及诱导有丝分裂细胞死亡。
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TAO Kinase inhibitor 1 是一种ATP 竞争性的thousand-and-one amino acid kinases (TAOK)选择性抑制剂,对于 TAOK1 和 TAOK2 的IC50s 分别为 11 nM 和 15 nM。它能够延迟有丝分裂以及诱导有丝分裂细胞死亡。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 285 | 现货 | |
5 mg | ¥ 652 | 现货 | |
10 mg | ¥ 996 | 现货 | |
25 mg | ¥ 2,180 | 现货 | |
50 mg | ¥ 3,430 | 现货 | |
100 mg | ¥ 4,990 | 现货 | |
500 mg | ¥ 10,500 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 721 | 现货 |
产品描述 | TAO Kinase inhibitor 1 delays mitosis and induces mitotic cell death. TAO Kinase inhibitor 1 is a selective and ATP-competitive thousand-and-one amino acid kinases inhibitor (IC50s: 11 to 15 nM for TAOK1 and 2, respectively). |
靶点活性 | TAOK2:15 nM, TAOK1:11 nM |
分子量 | 384.47 |
分子式 | C25H24N2O2 |
CAS No. | 850467-66-2 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 55 mg/mL (143.05 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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