购物车
  • 全部删除
  • TargetMol
    您的购物车当前为空
筛选
已筛选:全部清除
TargetMol | Tags 通过 Target 筛选
  • ADC Linker
    (1)
  • Antifection
    (1)
  • Antioxidant
    (1)
  • Drug Metabolite
    (2)
  • Estrogen Receptor/ERR
    (2)
  • IL Receptor
    (1)
  • MAO
    (1)
  • OX Receptor
    (1)
  • Others
    (145)
筛选
搜索结果
TargetMol产品目录中 "

estradiol 17-(b-d-glucuronide)

"的结果
  • 抑制剂&激动剂
    170
    TargetMol | Inhibitors_Agonists
  • 多肽产品
    4
    TargetMol | Peptide_Products
  • 染料试剂
    4
    TargetMol | Dye_Reagents
  • 天然产物
    36
    TargetMol | Natural_Products
  • 同位素
    4
    TargetMol | Isotope_Products
beta-Estradiol 17-hemisuccinatebeta-雌二醇 17-半琥珀酸酯
T96047698-93-3
beta-Estradiol 17-hemisuccinate 选择性染色富含雌激素受体 (ER) 的细胞。
  • ¥ 780
现货
规格
数量
TargetMol | Inhibitor Sale
6-Chloro-3-indolyl-β-D-Glucuronide CHA16beta-Methyl-16alpha,17alpha-epoxypregnenolone
T37811138182-20-4
6-Chloro-3-indolyl-β-D-Glucuronide (cyclohexylammonium salt) 是 β-glucuronidase 的显色底物。 6-Chloro-3-indolyl-β-D-Glucuronide (cyclohexylammonium salt) 可用于组织化学分析 β-glucuronidase 活性。
  • ¥ 113
现货
规格
数量
TargetMol | Inhibitor Sale
oroxylin A 7-O-β-d-glucuronide千层纸素A-7葡萄糖苷
TN678236948-77-3
oroxylin A 7-O-β-d-glucuronide 是一种新的生物碱,发现于石蒜的鳞茎中。
  • ¥ 772
现货
规格
数量
Pseudolaric acid B β-D-glucosidePseudolaric acid B-glucopyranoside,土槿皮乙酸-O-Β- D -葡萄糖苷,土荆皮乙酸苷
T574198891-41-9
Pseudolaric acid B β-D-glucoside (Pseudolaric acid B-glucopyranoside) 是一种二萜酸,分离自Pseudolarix kaempferi 中。
  • ¥ 186
现货
规格
数量
TargetMol | Inhibitor Sale
Glycyrrhetic acid 3-O-β-D-glucuronide单葡萄糖醛酸甘草次酸,Glycyrrhetic acid 3-O-mono-beta-D-glucuronide
TN170434096-83-8
Glycyrrhetic acid 3-O-mono-beta-D-glucuronide 是从甘草中分离出的甘草酸 3-O-β-D-葡萄糖醛酸,是甘草甜素的重要衍生物。它具有抗过敏活性,可作为甜味剂。
  • ¥ 442
现货
规格
数量
TargetMol | Inhibitor Sale
Torachrysone-8-O-b-D-glucosideTorachrysone 8-O-glucoside,芦荟大黄素 8-葡萄糖甙
TN227764032-49-1
Torachrysone-8-O-b-D-glucoside 可从 Polygonum multiflorum 分离得到。它对 DPCs(真皮乳头细胞)的增殖具有促进作用。
  • ¥ 1160
现货
规格
数量
TargetMol | Inhibitor Sale
β-Estradiol 17-acetateβ-雌二醇 17-乙酸酯,17-乙酸-17-BETA-雌二酯,beta-estradiol 17-acetate,1,3,5(10)-Estratriene-3,17β-diol 17-acetate
T72991743-60-8
β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) 是一种雌二醇代谢物。
  • ¥ 415
现货
规格
数量
TargetMol | Inhibitor Sale
MAO-B-IN-17
T607122890188-81-3
MAO-B-IN-17 是一种具有选择性和有效性的单胺氧化酶 B (MAO-B) 抑制剂(IC50:5.08 μM),可用于研究像帕金森类的中枢神经系统疾病。
  • ¥ 283
现货
规格
数量
Luteolin-3-O-beta-D-glucuronide木犀草素-3'-葡萄糖醛酸苷
TQ007053527-42-7
Luteolin-3-O-beta-D-glucuronide 是木犀草素葡萄糖醛酸,木犀草素的 3’ 端位置有 β-d-葡萄糖苷酸残基。
  • ¥ 628
现货
规格
数量
TargetMol | Inhibitor Sale
Kaempferol 3-O-β-D-glucuronideKaempferol-3-O-glucuronide,Kaempferol-3-beta-O-glucuronide,山奈酚葡萄糖醛酸苷,Kaempferol-3-glucuronide
TN181822688-78-4
Kaempferol 3-O-β-D-glucuronide (Kaempferol-3-beta-O-glucuronide) 具有抗氧化活性。 类黄酮葡糖苷酸可以被来自各种人体细胞的微粒体 α2-葡糖苷酸酶解偶联。
  • ¥ 955
现货
规格
数量
1,4-b-D-Xylopentaose木五糖,Xylopentaose
T816449694-20-4
1,4-b-D-Xylopentaose 是由 5 个b-1,4 木糖组成。
  • ¥ 529
现货
规格
数量
DiosMetin 7-O-β-D-Glucuronide
T1104735110-20-4
DiosMetin 7-O-β-D-Glucuronide 是一种丝瓜中的抗氧化成分。
  • ¥ 897
现货
规格
数量
TargetMol | Inhibitor Sale
Mycophenolic acid-β-D-glucuronide霉酸Β-D -葡萄糖醛酸溶液
T6010431528-44-6
Mycophenolic acid glucuronide 是人血浆中mycophenolic acid 的葡糖甙代谢产物。
  • ¥ 913
现货
规格
数量
TargetMol | Inhibitor Sale
[Ala11,D-Leu15]-Orexin B acetate[Ala11,D-Leu15]-Orexin B acetate (532932-99-3 Free base)
TP1975L
[Ala11,D-Leu15]-Orexin B acetate 是一种特异性 orexin-2 受体 (OX2) 激动剂,EC50 为 0.13 nM,比 OX1 (52 nM) 特异性高 400 倍。
  • ¥ 4497
现货
规格
数量
TargetMol | Inhibitor Sale
Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate)
T36807
Estradiol 17-(β-D-glucuronide) (E217G) is an estrogen metabolite formed in the liver and subsequently excreted in bile.1It acts as a substrate of the multidrug resistance protein 2 (MRP2; Km= 75 μM), and through MRP2-mediated transport, functions as a cholestatic agent, decreasing bile flow.1,2In addition to binding to the MRP2 transport site, E217G has been shown to bind to an allosteric site that through positive cooperativity activates its own transportviaMRP2 and the transport of other MRP2 substrates, including the non-cholestatic estrogen metabolite, estradiol 3-(β-D-glucuronide) .2,3E217G has also been reported to be transported by MDR1, MRP1, MRP3, MRP4, MRP7, ABCG2 (a breast cancer resistance protein transporter), and the rat organic anion-transporting polypeptides 1-4.2 1.Loe, D.W., Almquist, K.C., Cole, S.P., et al.ATP-dependent 17β-estradiol 17-(β-D-glucuronide) transport by multidrug resistance protein (MRP). Inhibition by cholestatic steroidsThe Journal of Biological Chemisty271(16)9683-9689(1996) 2.Gerk, P.M., Li, W., and Vore, M.Estradiol 3-glucuronide is transported by the multidrug resistance-associated protein 2 but does not activate the allosteric site bound by estradiol 17-glucuronideDrug Metabolism and Disposition32(10)1139-1145(2004) 3.Gerk, P.M., Li, W., Megaraj, W., et al.Human multidrug resistance protein 2 transports the therapeutic bile salt tauroursodeoxycholateJournal of Pharmacology and Experimental Therapeutics320(2)893-899(2007)
  • ¥ 1270
35日内发货
规格
数量
(S)-Ibuprofen acyl-β-D-glucuronide(S)-Ibuprofen glucuronide
T8536498649-76-4
(S)-Ibuprofen acyl-β-D-glucuronide ((S)-Ibuprofen glucuronide) 作为 S-布洛芬的一种酰基葡萄糖醛酸代谢产物,主要存在于肝脏中。该化合物广泛应用于研究 S-布洛芬的代谢过程及药代动力学,S-布洛芬为常用的非甾体抗炎药。
  • 询价
10-14周
规格
数量
Deferiprone O-β-D-glucuronide
T86179141675-48-1
Deferiprone O-β-D-glucuronide 为新型口服活性铁螯合剂,可有效降低β-地中海贫血患者的铁负荷。
  • 询价
10-14周
规格
数量
Isopentyl b-D-glucoside
T126225120671-07-0
Isopentyl b-D-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126225,CAS号为 120671-07-0。
  • ¥ 9995
6-8周
规格
数量
4-Amino-1-(b-D-ribofuranosyl)-7H-pyrrolo[2.3-d]pyrimidine-5-carboxamide
TNU0272
Nucleoside Derivatives - 7-Deaza-purine nucleosides; Natural product; inhibitor of protein kinase C 蛋白激酶抑制剂
  • 询价
5日内发货
规格
数量
4,6-Diamino-3-iodo-1-(b-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine
TNU0283908143-13-5
Nucleoside Derivatives - 8-Aza-7-deaza purine nucleosides, Halo-nucleosides
  • 询价
5日内发货
规格
数量
2’-Deoxy-2’-fluoro-b-D-arabino-6-azauridine
TNU0302908129-24-8
2'-Deoxy-2'-fluoro-b-D-arabino-6-azauridine is a Nucleoside Derivative - 6-Aza-uridine; Fluoro-modified nucleoside; Arabino nucleoside.
  • 询价
5日内发货
规格
数量
9-(b-D-Xylofuranosyl)guanine
TNU026727462-39-1
9-(b-D-Xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside.
  • 询价
5日内发货
规格
数量
1-Amino-7-cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl)guanine
TNU03872389988-22-9
Nucleoside Derivatives - Xylo-nucleosides; 8-Modified purine nucleosides; Amino nucleosides; N-Methylated alkylated nucleosides
  • 询价
5日内发货
规格
数量
(15aR)-1,15-Bis(diphenylphosphino)-7,8,9,10-tetrahydro-6H-dibenzo[b,d][1,6]dioxacycloundecine
T67391301847-91-6
(15aR)-1,15-Bis(diphenylphosphino)-7,8,9,10-tetrahydro-6H-dibenzo[b,d][1,6]dioxacycloundecine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67391。
  • 询价
5日内发货
规格
数量
Quercetin 3-O-(6-O-malonyl)-b-D-glucoside
T12383896862-01-0
Quercetin 3-O-(6-O-malonyl)-b-D-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T123838,CAS号为 96862-01-0。
  • 询价
规格
数量
1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine
TNU03852389988-20-7
1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside; 8-Modified purine nucleoside; Amino nucleoside.
  • 询价
5日内发货
规格
数量
6-Amino-3-iodo-4-methoxy-1-(b-D-ribofuranosyl)-1H-pyrazolo[3,4-d]pyrimidine
TNU02811997362-11-4
Nucleoside Derivatives - 7-Deaza-8-aza purine nucleosides; Halo-nucleosides; 6-Modified purine nucleosides
  • 询价
5日内发货
规格
数量
2-Amino-4-chloro-5-iodo-N2-pivaloyl-7-[2-deoxy-3,5-di-O- (4-methylbenzoyl)-b-D-ribofuanosyl]-7H-pyrrolo[2,3-d]pyrimidine
TNU1291199938-73-3
2-Amino-4-chloro-5-iodo-N2-pivaloyl-7-[2-deoxy-3,5-di-O- (4-methylbenzoyl)-b-D-ribofuanosyl]-7H-pyrrolo[2,3-d]pyrimidine is a Nucleoside Derivative - 7-Deazapurine nucleoside; Halo-nucleoside.
  • 询价
5日内发货
规格
数量
Tolmetin β-D-Glucuronide
T3612871595-19-2
Tolmetin β-D-Glucuronide 与人血清白蛋白具有反应特性,可通过串联质谱法鉴定结合位点和反应机制。
  • ¥ 4230
35日内发货
规格
数量
2’-Amino-2’-deoxy-b-D-arabino-5-methyl uridine
TNU0501135304-48-2
Nucleoside Derivatives - 2’-Modified nucleosides; Amino nucleosides
  • 询价
5日内发货
规格
数量
(R)-a-Terpinyl b-D-glucoside
T126338114673-99-3
(R)-a-Terpinyl b-D-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126338,CAS号为 114673-99-3。
  • 询价
规格
数量
N4-Benzoyl-2’-deoxy-2’-fluoro-b-D-arabinocytidine
TNU1174
N4-Benzoyl-2’-deoxy-2’-fluoro-b-D-arabinocytidine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TNU1174。
  • 询价
5日内发货
规格
数量
6-Methoxy-9-(3-deoxy-3-fluoro-b-D-ribofuranosyl)-9H-purine
TNU01542072145-35-6
Nucleoside Derivatives –Fluoro-modified nucleosides, 6-Modified purine nucleosides, 3’-Modified nucleosides
  • 询价
5日内发货
规格
数量
Propofol β-D-Glucuronide
T37378114991-26-3
Propofol β-D-glucuronide is a metabolite of propofol sulfate , a short-acting anesthetic agent. [1] [2] The metabolite is generated through the glucuronidation of propofol by uridine diphosphate glucuronosyltransferases. Propofol metabolism appears to occur more rapidly in women than men. [1]
  • ¥ 560
35日内发货
规格
数量
1-b-D-(3-Methoxy naphthalen-2-yl)-2’-deoxyriboside; 1,4-Anhydro-2-deoxy-1-C-(3-methoxy)-naphthalenyl)-D-erythro-pentitol
TNU16411117893-19-2
1-b-D-(3-Methoxy naphthalen-2-yl)-2’-deoxyriboside; 1,4-Anhydro-2-deoxy-1-C-(3-methoxy)-naphthalenyl)-D-erythro-pentitol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TNU1641,CAS号为 1117893-19-2。
  • 询价
5日内发货
规格
数量
2-Amino-4-chloro-N2-pivaloyl-7-[2-deoxy-3,5-di-O-(4- methylbenzoyl)-b-D-ribofuanosyl]-7H-pyrrolo[2,3-d]pyrimidine
TNU12901878120-03-6
2-Amino-4-chloro-N2-pivaloyl-7-[2-deoxy-3,5-di-O-(4- methylbenzoyl)-b-D-ribofuanosyl]-7H-pyrrolo[2,3-d]pyrimidine is a Nucleoside Derivative - 7-Deazapurine nucleoside; Halo-nucleoside.
  • 询价
5日内发货
规格
数量
1-(b-D-Xylofuranosyl)-N6-(p-methoxybenzyl)   adenine
TNU1485
1-(b-D-Xylofuranosyl)-N6-(p-methoxybenzyl) adenine is a Nucleoside Derivative - Xylo-nucleoside, 6-Modified purine nucleoside.
  • 询价
5日内发货
规格
数量
1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one
TNU08002072145-17-4
1-(2-C-b-Methyl-b-D-ribofuranosyl)-5-nitropyridine-2(1H)-one is a Pyridine nucleoside; 2'-C-Methyl nucleoside.
  • 询价
5日内发货
规格
数量
5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine
T644371265884-98-7
5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64437。
  • 询价
5日内发货
规格
数量
1-(b-D-Xylofuranosyl)-N6-(m-trifluoromethyl   benzyl) adenine
TNU0524
1-(b-D-Xylofuranosyl)-N6-(m-trifluoromethyl benzyl) adenine is a Nucleoside Derivative - Xylo-nucleoside, 6-Modified purine nucleoside, Fluoro-modified nucleoside.
  • 询价
5日内发货
规格
数量
(±)-4-hydroxy Propranolol β-D-Glucuronide
T3540294731-13-2
(±)-4-hydroxy Propranolol β-D-glucuronide is a metabolite of (±)-4-hydroxy propranolol , which is a metabolite of propranolol. The apparent half-life of (±)-4-hydroxy propranolol β-D-glucuronide is similar to propranolol and 4-hydroxy propranolol. Propranolol is a β-adrenergic antagonist, and the active enantiomer, (S)-(-)-propranolol , has log Kd values of -8.16, -9.08, and -6.93 for β1, β2, and β3, respectively.
  • ¥ 2970
35日内发货
规格
数量
7-(2-Deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine
TNU103293366-89-3
Nucleoside Derivatives - 7-Deaza-purine nucleosides; 6-De-aminopurine nucleosides
  • 询价
5日内发货
规格
数量
1-(b-D-Xylofuranosyl)-2-thiouracil
TNU03712305416-17-3
Nucleoside Derivatives - Xylo-nucleosides, Thio-nucleosides
  • 询价
5日内发货
规格
数量
2’-Deoxy-2’-fluoro-4’-thio-b-D-arabinouridine
TNU0518941610-00-0
2'-Deoxy-2'-fluoro-4'-thio-b-D-arabinouridine is a Nucleoside Derivative - Thio-nucleoside;Fluoro-modified -nucleoside.
  • 询价
5日内发货
规格
数量
Naringenin-7-O-β-D-Glucuronide
TN72621237479-07-0
Naringenin-7-O-β-D-glucuronide, a metabolite of the flavonoid naringenin, is predominantly synthesized through the action of UDP-glucuronosyltransferase (UGT) isoforms UGT1A1, UGT1A3, UGT1A6, and UGT1A9.
  • 询价
规格
数量
Cyclobenzaprine b-D-glucuronide环苯扎林-N-葡萄糖醛酸
T8860167324-97-4
Cyclobenzaprine b-D-glucuronide,作为Cyclobenzaprine的代谢产物,具有治疗冠状病毒(Coronavirus)相关疾病的潜力。此外,还可用于研究Cyclobenzaprine在体内的代谢路径,以及作为研究冠状病毒治疗潜在候选物的重要工具。
  • 询价
10-14周
规格
数量
Ichangin-4-O-b-D-glucopyranoside
T126082129502-62-1
Ichangin-4-O-b-D-glucopyranoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126082,CAS号为 129502-62-1。
  • 询价
规格
数量